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Binding of cardiotonic steroids to Na(+),K(+)-ATPase in the E2P state

The sodium pump (Na(+), K(+)-ATPase, NKA) is vital for animal cells, as it actively maintains Na(+) and K(+) electrochemical gradients across the cell membrane. It is a target of cardiotonic steroids (CTSs) such as ouabain and digoxin. As CTSs are almost unique strong inhibitors specific to NKA, a w...

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Dades bibliogràfiques
Publicat a:Proc Natl Acad Sci U S A
Autors principals: Kanai, Ryuta, Cornelius, Flemming, Ogawa, Haruo, Motoyama, Kanna, Vilsen, Bente, Toyoshima, Chikashi
Format: Artigo
Idioma:Inglês
Publicat: National Academy of Sciences 2021
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7817145/
https://ncbi.nlm.nih.gov/pubmed/33318128
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.2020438118
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