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Automated, Accurate, and Scalable Relative Protein-Ligand Binding Free Energy Calculations using Lambda Dynamics

Accurate predictions of changes to protein-ligand binding affinity in response to chemical modifications are of utility in small molecule lead optimization. Relative free energy perturbation (FEP) approaches are one of the most widely utilized for this goal, but involve significant computational cos...

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Vydáno v:J Chem Theory Comput
Hlavní autoři: Raman, E. Prabhu, Paul, Thomas J., Hayes, Ryan L., Brooks, Charles L.
Médium: Artigo
Jazyk:Inglês
Vydáno: 2020
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC7814773/
https://ncbi.nlm.nih.gov/pubmed/33201701
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jctc.0c00830
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