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Direct synthesis of anomeric tetrazolyl iminosugars from sugar-derived lactams

Herein we present the direct asymmetric synthesis of tetrazole-functionalized 1-deoxynojirimycin derivatives from simple sugars via a Schwartz’s reagent-mediated reductive amide functionalization followed by a variant of the Ugi–azide multicomponent reaction. The anomeric configurations of two produ...

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Detaylı Bibliyografya
Yayımlandı:Beilstein J Org Chem
Asıl Yazarlar: Więcław, Michał Mateusz, Furman, Bartłomiej
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: Beilstein-Institut 2021
Konular:
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC7814180/
https://ncbi.nlm.nih.gov/pubmed/33519998
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3762/bjoc.17.12
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