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Transient States and Barriers from Molecular Simulations and the Milestoning Theory: Kinetics in Ligand–Protein Recognition and Compound Design

This study presents a novel computational approach to study molecular recognition and binding kinetics for drug-like compounds dissociating from a flexible protein system. The intermediates and their free energy profile during ligand association and dissociation processes control ligand–protein bind...

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Publicado en:J Chem Theory Comput
Autores principales: Tang, Zhiye, Chen, Si-Han, Chang, Chia-en A.
Formato: Artigo
Lenguaje:Inglês
Publicado: 2020
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC7809013/
https://ncbi.nlm.nih.gov/pubmed/32031801
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jctc.9b01153
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