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Prediction of kinase inhibitors binding modes with machine learning and reduced descriptor sets

Protein kinases are receiving wide research interest, from drug perspective, due to their important roles in human body. Available kinase-inhibitor data, including crystallized structures, revealed many details about the mechanism of inhibition and binding modes. The understanding and analysis of th...

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Bibliografski detalji
Izdano u:Sci Rep
Glavni autori: Abdelbaky, Ibrahim, Tayara, Hilal, Chong, Kil To
Format: Artigo
Jezik:Inglês
Izdano: Nature Publishing Group UK 2021
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC7804204/
https://ncbi.nlm.nih.gov/pubmed/33436888
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41598-020-80758-4
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