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Farnesyl Transferase Inhibitor Lonafarnib Enhances α7nAChR Expression Through Inhibiting DNA Methylation of CHRNA7 and Increases α7nAChR Membrane Trafficking

Inhibition of Ras farnesylation in acute has been found to upregulate the α7 nicotinic acetylcholine receptor (α7nAChR) activity. This study was carried out to investigate the effect of chronic administration for 7 days of farnesyl transferase inhibitor lonafarnib (50 mg/kg, intraperitoneally inject...

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Publicat a:Front Pharmacol
Autors principals: Chen, Tingting, Cai, Chengyun, Wang, Lifeng, Li, Shixin, Chen, Ling
Format: Artigo
Idioma:Inglês
Publicat: Frontiers Media S.A. 2020
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7801264/
https://ncbi.nlm.nih.gov/pubmed/33447242
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3389/fphar.2020.589780
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