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Cyclic peptides: Backbone rigidification and capability of mimicking motifs at protein–protein interfaces

Cyclization is commonly employed in efforts to improve the target binding affinity of peptide-based probes and therapeutics. Many structural motifs have been identified at protein–protein interfaces and provide promising targets for inhibitor design using cyclic peptides. Cyclized peptides are gener...

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Publicat a:Phys Chem Chem Phys
Autors principals: Huang, He, Damjanovic, Jovan, Miao, Jiayuan, Lin, Yu-Shan
Format: Artigo
Idioma:Inglês
Publicat: 2021
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7790991/
https://ncbi.nlm.nih.gov/pubmed/33331371
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/d0cp04633g
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