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Design of a multivalent bifunctional chelator for diagnostic (64)Cu PET imaging in Alzheimer’s disease

Herein, we report a (64)Cu positron emission tomography (PET) imaging agent that shows appreciable in vivo brain uptake and exhibits high specific affinity for beta-amyloid (Aβ) aggregates, leading to the successful PET imaging of amyloid plaques in the brains of 5xFAD mice versus those of wild-type...

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Pubblicato in:Proc Natl Acad Sci U S A
Autori principali: Cho, Hong-Jun, Huynh, Truc T., Rogers, Buck E., Mirica, Liviu M.
Natura: Artigo
Lingua:Inglês
Pubblicazione: National Academy of Sciences 2020
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7733815/
https://ncbi.nlm.nih.gov/pubmed/33234563
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.2014058117
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