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Drug-like properties in macrocycles above MW 1000: Backbone rigidity vs. side-chain lipophilicity

Large, macrocyclic peptides can achieve surprisingly high membrane permeability, although the properties that govern permeability in this chemical space are only beginning to come into focus. We generated two libraries of cyclic decapeptides with stable, cross-β conformations, and found that peptoid...

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Detalhes bibliográficos
Publicado no:Angew Chem Int Ed Engl
Main Authors: Furukawa, Akihiro, Schwochert, Joshua, Pye, Cameron R., Asano, Daigo, Edmondson, Quinn D., Turmon, Alexandra C., Klein, Victoria G., Ono, Satoshi, Okada, Okimasa, Lokey, R. Scott
Formato: Artigo
Idioma:Inglês
Publicado em: 2020
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7719619/
https://ncbi.nlm.nih.gov/pubmed/32789999
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/anie.202004550
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