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Developing a Kinase-Specific Target Selection Method Using a Structure-Based Machine Learning Approach

INTRODUCTION: Despite recent advances in the drug discovery field, developing selective kinase inhibitors remains a complicated issue for a number of reasons, one of which is that there are striking structural similarities in the ATP-binding pockets of kinases. OBJECTIVE: To address this problem, we...

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Pubblicato in:Adv Appl Bioinform Chem
Autori principali: Afanasyeva, Arina, Nagao, Chioko, Mizuguchi, Kenji
Natura: Artigo
Lingua:Inglês
Pubblicazione: Dove 2020
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7719317/
https://ncbi.nlm.nih.gov/pubmed/33293834
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.2147/AABC.S278900
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