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MODL-17. SHP2 INHIBITORS SHOW ACTIVITY AGAINST NF1-DEFICIENT GLIOMAS AND ENHANCE MAPK PATHWAY INHIBITION IN BRAF-V600E MUTANT GLIOMAS

INTRODUCTION: Activation of the RAS-MAPK signaling cascade is common in pediatric gliomas. Based on the role of SHP2 in RAS pathway signaling, we hypothesized that NF1-deficient pediatric glioma models would respond to SHP2 inhibitor monotherapy whereas BRAF-V600E gliomas would not. However, we post...

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Bibliografski detalji
Izdano u:Neuro Oncol
Glavni autori: Muldoon, Daniel, Zhao, Guisheng, Batt, Carly, Singh, Mallika, Nicolaides, Theodore
Format: Artigo
Jezik:Inglês
Izdano: Oxford University Press 2020
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC7715749/
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1093/neuonc/noaa222.591
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