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PCSK9 Inhibition: Insights From Clinical Trials and Future Prospects

In 2003, clinical observations led to the discovery of the involvement of proprotein convertase subtilisin/kexin type 9 (PCSK9) in lipid metabolism. Functional studies demonstrated that PCSK9 binds to the low-density lipoprotein (LDL) receptor directing it to its lysosomal degradation. Therefore, ca...

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Publicado en:Front Physiol
Main Authors: Katzmann, Julius L., Gouni-Berthold, Ioanna, Laufs, Ulrich
Formato: Artigo
Idioma:Inglês
Publicado: Frontiers Media S.A. 2020
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC7701092/
https://ncbi.nlm.nih.gov/pubmed/33304274
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3389/fphys.2020.595819
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