Homologation of the Fischer Indolization: A Quinoline Synthesis via Homo‐Diaza‐Cope Rearrangement

We disclose a new Brønsted acid promoted quinoline synthesis, proceeding via homo‐diaza‐Cope rearrangement of N‐aryl‐N′‐cyclopropyl hydrazines. Our strategy can be considered a homologation of Fischer's classical indole synthesis and delivers 6‐membered N‐heterocycles, including previously inac...

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Dades bibliogràfiques
Publicat a:Angew Chem Int Ed Engl
Autors principals: Gerosa, Gabriela Guillermina, Schwengers, Sebastian Armin, Maji, Rajat, De, Chandra Kanta, List, Benjamin
Format: Artigo
Idioma:Inglês
Publicat: John Wiley and Sons Inc. 2020
Matèries:
Communications
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7693176/
https://ncbi.nlm.nih.gov/pubmed/32621795
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/anie.202005798
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