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Domain-Swap Dimerization of Acanthamoeba castellanii CYP51 and a Unique Mechanism of Inactivation by Isavuconazole

Cytochromes P450 (P450, CYP) metabolize a wide variety of endogenous and exogenous lipophilic molecules, including most drugs. Sterol 14α-demethylase (CYP51) is a target for antifungal drugs known as conazoles. Using X-ray crystallography, we have discovered a domain-swap homodimerization mode in CY...

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Detaylı Bibliyografya
Yayımlandı:Mol Pharmacol
Asıl Yazarlar: Sharma, Vandna, Shing, Brian, Hernandez-Alvarez, Lilian, Debnath, Anjan, Podust, Larissa M.
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: The American Society for Pharmacology and Experimental Therapeutics 2020
Konular:
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC7674934/
https://ncbi.nlm.nih.gov/pubmed/33008918
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/molpharm.120.000092
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