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Deazaflavin inhibitors of TDP2 with cellular activity can affect etoposide influx and/or efflux

Tyrosyl DNA phosphodiesterase 2 (TDP2) facilitates the repair of topoisomerase II (TOP2)-linked DNA double-strand breaks and as a consequence is required for cellular resistance to TOP2 “poisons”. Recently, a deazaflavin series of compounds were identified as potent inhibitors of TDP2, in vitro. Her...

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Bibliografiske detaljer
Udgivet i:ACS Chem Biol
Main Authors: Komulainen, Emilia, Pennicott, Lewis, Grand, Darren Le, Caldecott, Keith W
Format: Artigo
Sprog:Inglês
Udgivet: 2019
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC7613159/
https://ncbi.nlm.nih.gov/pubmed/31091068
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acschembio.9b00144
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