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Recent advances in the design of RAR α and RAR β agonists as orally bioavailable drugs. A review

Retinoic acid receptors (RARs) α, β, and γ are members of the nuclear receptor superfamily. Compounds which bind to and activate the RARs are termed retinoids which regulate a wide variety of biological processes such as vertebrate embryonic morphogenesis and organogenesis, cell growth arrest, diffe...

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Publicat a:Bioorg Med Chem
Autors principals: Borthwick, Alan D., Goncalves, Maria B., Corcoran, Jonathan P.T.
Format: Artigo
Idioma:Inglês
Publicat: Elsevier Science 2020
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7588594/
https://ncbi.nlm.nih.gov/pubmed/33069074
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2020.115664
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