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Amphiphilic Aminoglycosides as Medicinal Agents

The conjugation of hydrophobic group(s) to the polycationic hydrophilic core of the antibiotic drugs aminoglycosides (AGs), targeting ribosomal RNA, has led to the development of amphiphilic aminoglycosides (AAGs). These drugs exhibit numerous biological effects, including good antibacterial effects...

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Dettagli Bibliografici
Pubblicato in:Int J Mol Sci
Autori principali: Dezanet, Clément, Kempf, Julie, Mingeot-Leclercq, Marie-Paule, Décout, Jean-Luc
Natura: Artigo
Lingua:Inglês
Pubblicazione: MDPI 2020
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7583001/
https://ncbi.nlm.nih.gov/pubmed/33049963
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ijms21197411
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