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Computing ligands bound to proteins using MELD-accelerated MD

Predicting the poses of small-molecule ligands in protein binding sites is often done by virtual screening algorithms like DOCK. In principle, Molecular Dynamics (MD) using atomistic force fields could give better free-energy-based pose selection, but MD is computationally expensive. Here, we ask if...

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Pubblicato in:J Chem Theory Comput
Autori principali: Liu, Cong, Brini, Emiliano, Perez, Alberto, Dill, Ken A.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2020
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7572789/
https://ncbi.nlm.nih.gov/pubmed/32910647
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jctc.0c00543
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