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DPAGT1 Inhibitors of Capuramycin Analogues and Their Antimigratory Activities of Solid Tumors

Capuramycin displays narrow spectrum of antibacterial activity by targeting bacterial translocase I (MraY). In our program of development of new N-acetylglucosaminephosphotransferase1 (DPAGT1) inhibitor, we have identified that a capuramycin phenoxypiperidinylbenzylamide analogue (CPPB) inhibits DPA...

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Detalhes bibliográficos
Publicado no:J Med Chem
Main Authors: Mitachi, Katsuhiko, Kansal, Rita G., Hevener, Kirk E., Gillman, Cody D., Hussain, Syed M., Yun, Hyun Gi, Miranda-Carboni, Gustavo A., Glazer, Evan S., Clemons, William M., Kurosu, Michio
Formato: Artigo
Idioma:Inglês
Publicado em: 2020
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7554145/
https://ncbi.nlm.nih.gov/pubmed/32886511
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.0c00545
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