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Mechanistic Insights into the Activation of Ester Prodrugs of 666-15

cAMP-response element binding protein (CREB) is an oncogenic transcription factor implicated in many different types of cancer. We previously reported the discovery of 666-15 as a potent inhibitor of CREB-mediated gene transcription. In an effort to improve the aqueous solubility of 666-15, amino es...

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Detalles Bibliográficos
Publicado en:Bioorg Med Chem Lett
Main Authors: Xie, Fuchun, Martin-Acosta, Pedro, Li, Bingbing X., Xiao, Xiangshu
Formato: Artigo
Idioma:Inglês
Publicado: 2020
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC7530057/
https://ncbi.nlm.nih.gov/pubmed/32730943
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2020.127455
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