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Identification, Synthesis and Evaluation of Substituted Benzofurazans as Inhibitors of CREB-mediated Gene Transcription

Cyclic-AMP response-element binding protein (CREB) is a stimulus-activated transcription factor. Its transcription activity requires its binding with CREB-binding protein (CBP) after CREB is phosphorylated at Ser133. The domains involved for CREB-CBP interaction are kinase-inducible domain (KID) fro...

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Detalhes bibliográficos
Main Authors: Xie, Fuchun, Li, Bingbing X., Broussard, Candice, Xiao, Xiangshu
Formato: Artigo
Idioma:Inglês
Publicado em: 2013
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3783659/
https://ncbi.nlm.nih.gov/pubmed/23953193
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2013.07.053
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