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Allosteric Mechanisms of Nonadditive Substituent Contributions to Protein-Ligand Binding

Quantifying chemical substituent contributions to ligand-binding free energies is challenging due to nonadditive effects. Protein allostery is a frequent cause of nonadditivity, but the underlying allosteric mechanisms often remain elusive. Here, we propose a general NMR-based approach to elucidate...

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書目詳細資料
發表在:Biophys J
Main Authors: Boulton, Stephen, Van, Katherine, VanSchouwen, Bryan, Augustine, Jerry, Akimoto, Madoka, Melacini, Giuseppe
格式: Artigo
語言:Inglês
出版: The Biophysical Society 2020
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在線閱讀:https://ncbi.nlm.nih.gov/pmc/articles/PMC7499118/
https://ncbi.nlm.nih.gov/pubmed/32882185
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bpj.2020.07.038
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