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BETting on next-generation bromodomain inhibitors

Within the last decade, bromodomain and extraterminal (BET) domain inhibitors were introduced as the first in a wave of new agents known as bromodomain inhibitors. These original examples exhibited anti-inflammatory and anticancer properties, and some have progressed to human clinical trials. BET pr...

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Pubblicato in:Am J Clin Exp Urol
Autori principali: Collins, Matthew K, Chau, Cindy H, Price, Douglas K, Figg, William D
Natura: Artigo
Lingua:Inglês
Pubblicazione: e-Century Publishing Corporation 2020
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7486540/
https://ncbi.nlm.nih.gov/pubmed/32929408
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