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BET bromodomain inhibitors—A novel epigenetic approach in castration-resistant prostate cancer

The androgen receptor (AR) is central to the initiation and progression of prostate cancer, even after castration. There has been some success in therapies targeting AR signaling which have been shown to extend survival in men with castration-resistant prostate cancer (CRPC). However, durable respon...

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Publicat a:Cancer Biol Ther
Autors principals: Lochrin, Sarah E, Price, Douglas K, Figg, William D
Format: Artigo
Idioma:Inglês
Publicat: Taylor & Francis 2014
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC4622075/
https://ncbi.nlm.nih.gov/pubmed/25535892
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.4161/15384047.2014.962297
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