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Comparative Clinical Pharmacokinetics and Pharmacodynamics of HIV-1 Integrase Strand Transfer Inhibitors: An Updated Review

Bictegravir (BIC), cabotegravir (CAB), dolutegravir (DTG), elvitegravir (EVG) and raltegravir (RAL), are members of latest class of antiretrovirals (ARV) available to treat human immunodeficiency virus (HIV) infection, the integrase strand transfer inhibitors (INSTI). INSTIs are potent inhibitors of...

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Publicat a:Clin Pharmacokinet
Autors principals: Podany, Anthony T., Scarsi, Kimberly K., Pham, Michelle M., Fletcher, Courtney V.
Format: Artigo
Idioma:Inglês
Publicat: 2020
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7484053/
https://ncbi.nlm.nih.gov/pubmed/32462541
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s40262-020-00898-8
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