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AZD9291 inactivates the PRC2 complex to mediate tumor growth inhibition

Deregulated Polycomb repressive complex 2 (PRC2) is intimately involved in tumorigenesis and progression, making it an invaluable target for epigenetic cancer therapy. Disrupting the EZH2–EED interaction, which is required for PRC2 enzymatic activity, is a promising strategy for cancer treatment. Ho...

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Dettagli Bibliografici
Pubblicato in:Acta Pharmacol Sin
Autori principali: Zhang, Kai-li, Shen, Qian-qian, Fang, Yan-fen, Sun, Yi-ming, Ding, Jian, Chen, Yi
Natura: Artigo
Lingua:Inglês
Pubblicazione: Springer Singapore 2019
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7468275/
https://ncbi.nlm.nih.gov/pubmed/31171828
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41401-019-0248-2
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