A carregar...

The Enzyme‐Free Release of Nucleotides from Phosphoramidates Depends Strongly on the Amino Acid

Phosphoramidates composed of an amino acid and a nucleotide analogue are critical metabolites of prodrugs, such as remdesivir. Hydrolysis of the phosphoramidate liberates the nucleotide, which can then be phosphorylated to become the pharmacologically active triphosphate. Enzymatic hydrolysis has be...

ver descrição completa

Na minha lista:
Detalhes bibliográficos
Publicado no:Angew Chem Int Ed Engl
Main Authors: Jovanovic, Dejana, Tremmel, Peter, Pallan, Pradeep S., Egli, Martin, Richert, Clemens
Formato: Artigo
Idioma:Inglês
Publicado em: John Wiley and Sons Inc. 2020
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7436718/
https://ncbi.nlm.nih.gov/pubmed/32757352
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/anie.202008665
Tags: Adicionar Tag
Sem tags, seja o primeiro a adicionar uma tag!