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Picomolar Affinity Antagonist and Sustained Signaling Agonist Peptide Ligands for the Adrenomedullin and Calcitonin Gene-Related Peptide Receptors

[Image: see text] The calcitonin receptor-like class B G protein-coupled receptor (CLR) mediates adrenomedullin (AM) and calcitonin gene-related peptide (CGRP) functions including vasodilation, cardioprotection, and nociception. Receptor activity-modifying proteins (RAMP1–3) form heterodimers with C...

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Publicado en:ACS Pharmacol Transl Sci
Autores principales: Booe, Jason M., Warner, Margaret L., Pioszak, Augen A.
Formato: Artigo
Lenguaje:Inglês
Publicado: American Chemical Society 2020
Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC7432658/
https://ncbi.nlm.nih.gov/pubmed/32832875
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsptsci.0c00031
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