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Probing the Plasticity in the Active Site of Protein N-terminal Methyltransferase 1 Using Bisubstrate Analogs

The bisubstrate analog strategy is a promising approach to develop potent and selective inhibitors for protein methyltransferases. Herein, the interactions of a series of bisubstrate analogs with protein N-terminal methyltransferase 1 (NTMT1) were examined to probe the molecular properties of the NT...

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Pubblicato in:J Med Chem
Autori principali: Chen, Dongxing, Dong, Cheng, Dong, Guangping, Srinivasan, Karthik, Min, Jinrong, Noinaj, Nicholas, Huang, Rong
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2020
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7429357/
https://ncbi.nlm.nih.gov/pubmed/32605369
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.0c00770
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