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Instability of aquaglyceroporin (AQP) 2 contributes to drug resistance in Trypanosoma brucei

Defining mode of action is vital for both developing new drugs and predicting potential resistance mechanisms. Sensitivity of African trypanosomes to pentamidine and melarsoprol is predominantly mediated by aquaglyceroporin 2 (TbAQP2), a channel associated with water/glycerol transport. TbAQP2 is ex...

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Dades bibliogràfiques
Publicat a:PLoS Negl Trop Dis
Autors principals: Quintana, Juan F., Bueren-Calabuig, Juan, Zuccotto, Fabio, de Koning, Harry P., Horn, David, Field, Mark C.
Format: Artigo
Idioma:Inglês
Publicat: Public Library of Science 2020
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7413563/
https://ncbi.nlm.nih.gov/pubmed/32644992
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1371/journal.pntd.0008458
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