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Unexpected Enhancement of HDACs Inhibition by MeS Substitution at C-2 Position of Fluoro Largazole

Given our previous finding that fluorination at the C18 position of largazole showed reasonably good tolerance towards inhibitory activity and selectivity of histone deacetylases (HDACs), further modification on the valine residue in the fluoro-largazole’s macrocyclic moiety with S-Me l-Cysteine or...

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Detalhes bibliográficos
Publicado no:Mar Drugs
Main Authors: Zhang, Bingbing, Ruan, Zhu-Wei, Luo, Dongdong, Zhu, Yueyue, Ding, Tingbo, Sui, Qiang, Lei, Xinsheng
Formato: Artigo
Idioma:Inglês
Publicado em: MDPI 2020
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7401273/
https://ncbi.nlm.nih.gov/pubmed/32629787
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/md18070344
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