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Comparative Assessment of Protein Kinase Inhibitors in Public Databases and in PKIDB

Since the first approval of a protein kinase inhibitor (PKI) by the Food and Drug Administration (FDA) in 2001, 55 new PKIs have reached the market, and many inhibitors are currently being evaluated in clinical trials. This is a clear indication that protein kinases still represent major drug target...

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Dettagli Bibliografici
Pubblicato in:Molecules
Autori principali: Bournez, Colin, Carles, Fabrice, Peyrat, Gautier, Aci-Sèche, Samia, Bourg, Stéphane, Meyer, Christophe, Bonnet, Pascal
Natura: Artigo
Lingua:Inglês
Pubblicazione: MDPI 2020
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7397241/
https://ncbi.nlm.nih.gov/pubmed/32679723
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules25143226
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