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2-Aminooxazole as a Novel Privileged Scaffold in Antitubercular Medicinal Chemistry

[Image: see text] To obtain effective eradication of numerous infectious diseases such as tuberculosis, it is important to supply the medicinal chemistry arsenal with novel chemical agents. Isosterism and bioisosterism are widely known concepts in the field of early drug discovery, and in several ca...

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Publicat a:ACS Med Chem Lett
Autors principals: Azzali, Elisa, Girardini, Miriam, Annunziato, Giannamaria, Pavone, Marialaura, Vacondio, Federica, Mori, Giorgia, Pasca, Maria Rosalia, Costantino, Gabriele, Pieroni, Marco
Format: Artigo
Idioma:Inglês
Publicat: American Chemical Society 2020
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7357219/
https://ncbi.nlm.nih.gov/pubmed/32676151
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsmedchemlett.0c00173
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