Elucidation of Inverse Agonist Activity of Bilastine

H(1)-antihistamines antagonize histamine and prevent it from binding to the histamine H(1) receptor (H1R). Some of them also act as inverse agonists, which are more potent than pure antagonists because they suppress the constitutive H1R activity. Bilastine is a non-sedative antihistamine which is on...

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Vydáno v:Pharmaceutics
Hlavní autoři: Mizuguchi, Hiroyuki, Wakugawa, Tomoharu, Sadakata, Hisato, Kamimura, Seiichiro, Takemoto, Mai, Nakagawa, Tomomi, Yabumoto, Masami, Kitamura, Yoshiaki, Takeda, Noriaki, Fukui, Hiroyuki
Médium: Artigo
Jazyk:Inglês
Vydáno: MDPI 2020
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Article
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC7355758/
https://ncbi.nlm.nih.gov/pubmed/32521742
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/pharmaceutics12060525
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