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Elucidation of Inverse Agonist Activity of Bilastine

H(1)-antihistamines antagonize histamine and prevent it from binding to the histamine H(1) receptor (H1R). Some of them also act as inverse agonists, which are more potent than pure antagonists because they suppress the constitutive H1R activity. Bilastine is a non-sedative antihistamine which is on...

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Detalhes bibliográficos
Publicado no:Pharmaceutics
Main Authors: Mizuguchi, Hiroyuki, Wakugawa, Tomoharu, Sadakata, Hisato, Kamimura, Seiichiro, Takemoto, Mai, Nakagawa, Tomomi, Yabumoto, Masami, Kitamura, Yoshiaki, Takeda, Noriaki, Fukui, Hiroyuki
Formato: Artigo
Idioma:Inglês
Publicado em: MDPI 2020
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7355758/
https://ncbi.nlm.nih.gov/pubmed/32521742
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/pharmaceutics12060525
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