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The arylstibonic acid compound NSC13746 disrupts B-ZIP binding to DNA in living cells

The inhibition of DNA binding of basic leucine zipper (B-ZIP) transcription factors is a clinically relevant molecular target. Our laboratory has previously reported two methods of inhibiting B-ZIP DNA binding in solution: 1) an arylstibonic acid compound that binds to the basic region, stabilizes t...

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Pubblicato in:Eur J Cell Biol
Autori principali: Heyerdahl, Sarah L., Rozenberg, Julian, Jamtgaard, Louis, Rishi, Vikas, Varticovski, Lyuba, Akah, Kelly, Scudiero, Dominic, Shoemaker, Robert H., Karpova, Tatiana S., Day, Richard N., McNally, James G., Vinson, Charles
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2010
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7316388/
https://ncbi.nlm.nih.gov/pubmed/20362353
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.ejcb.2009.11.029
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