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On Restraints in End-Point Protein-Ligand Binding Free Energy Calculations

The impact of harmonic restraints on protein heavy atoms and ligand atoms on end-point free energy calculations is systematically characterized for 54 protein-ligand complexes. We observe that stronger restraints reduce the equilibration time and statistical inefficiency, suppress conformational sam...

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Détails bibliographiques
Publié dans:J Comput Chem
Auteurs principaux: Menzer, William M., Xie, Bing, Minh, David D. L.
Format: Artigo
Langue:Inglês
Publié: 2019
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC7311925/
https://ncbi.nlm.nih.gov/pubmed/31821590
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/jcc.26119
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