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Dual orexin receptor antagonists increase sleep and cataplexy in wild type mice

Orexin receptor antagonists are clinically useful for treating insomnia, but thorough blockade of orexin signaling could cause narcolepsy-like symptoms. Specifically, while sleepiness is a desirable effect, an orexin antagonist could also produce cataplexy, sudden episodes of muscle weakness often t...

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Detalhes bibliográficos
Publicado no:Sleep
Main Authors: Mahoney, Carrie E, Mochizuki, Takatoshi, Scammell, Thomas E
Formato: Artigo
Idioma:Inglês
Publicado em: Oxford University Press 2019
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7294412/
https://ncbi.nlm.nih.gov/pubmed/31830270
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1093/sleep/zsz302
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