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PTC-174, a positive allosteric modulator of NMDA receptors containing GluN2C or GluN2D subunits

NMDA receptors are ionotropic glutamate receptors that mediate excitatory neurotransmission. The diverse functions of these receptors are tuned by deploying different combinations of GluN1 and GluN2 subunits (GluN2A-D) to form either diheteromeric NMDA receptors, which contain two GluN1 and two iden...

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Dettagli Bibliografici
Pubblicato in:Neuropharmacology
Autori principali: Yi, Feng, Rouzbeh, Nirvan, Hansen, Kasper B., Xu, Yuelian, Fanger, Christopher M., Gordon, Earl, Paschetto, Kathy, Menniti, Frank S., Volkmann, Robert A.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2020
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7293934/
https://ncbi.nlm.nih.gov/pubmed/31987864
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.neuropharm.2020.107971
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