Caricamento...

ABCG2 Deficiency Does Not Alter Dolutegravir Metabolism and Pharmacokinetics

Dolutegravir (DTG) is a potent integrase inhibitor of human immunodeficiency virus. Because DTG is a substrate of the efflux transporter ABCG2 and ABCG2 is highly polymorphic, we asked whether dose adjustment of DTG is needed for ABCG2-deficient individuals. Using Abcg2-null mice, the current work i...

Descrizione completa

Salvato in:
Dettagli Bibliografici
Pubblicato in:J Pharmacol Exp Ther
Autori principali: Zhu, Junjie, Tian, Xin, Shehu, Amina I., McMahon, Deborah K., Ma, Xiaochao
Natura: Artigo
Lingua:Inglês
Pubblicazione: The American Society for Pharmacology and Experimental Therapeutics 2020
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7292963/
https://ncbi.nlm.nih.gov/pubmed/32303561
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/jpet.119.264424
Tags: Aggiungi Tag
Nessun Tag, puoi essere il primo ad aggiungerne! !