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Development of a Cell-Permeable Cyclic Peptidyl Inhibitor against the Keap1-Nrf2 Interaction

Macrocyclic peptides have proven highly effective inhibitors of protein–protein interactions, but generally lack cell permeability to access intracellular targets. We show herein that macrocyclic peptides may be rendered highly cell-permeable and biologically active by conjugating with a cyclic cell...

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Pubblicato in:J Org Chem
Autori principali: Salim, Heba, Song, Jian, Sahni, Ashweta, Pei, Dehua
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2019
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7288753/
https://ncbi.nlm.nih.gov/pubmed/31609620
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.joc.9b02367
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