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The Use of Computational Approaches in the Discovery and Mechanism Study of Opioid Analgesics

Opioid receptors that belong to class A G protein-coupled receptors (GPCRs) are vital in pain control. In the past few years, published high-resolution crystal structures of opioid receptor laid a solid basis for both experimental and computational studies. Computer-aided drug design (CADD) has been...

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Publicat a:Front Chem
Autors principals: Zhao, Bangyi, Li, Wei, Sun, Lijie, Fu, Wei
Format: Artigo
Idioma:Inglês
Publicat: Frontiers Media S.A. 2020
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7242749/
https://ncbi.nlm.nih.gov/pubmed/32500054
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3389/fchem.2020.00335
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