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Novel and Modified Neutrophil Elastase Inhibitor Loaded in Topical Formulations for Psoriasis Management

Human neutrophil elastase (HNE) is a serine protease that degrades matrix proteins. An excess of HNE may trigger several pathological conditions, such as psoriasis. In this work, we aimed to synthesize, characterize and formulate new HNE inhibitors with a 4-oxo-β-lactam scaffold with less toxicity,...

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Kaydedildi:
Detaylı Bibliyografya
Yayımlandı:Pharmaceutics
Asıl Yazarlar: Nunes, Andreia, Marto, Joana, Gonçalves, Lídia Maria, Simões, Sandra, Félix, Rita, Ascenso, Andreia, Lopes, Francisca, Ribeiro, Helena Margarida
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: MDPI 2020
Konular:
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC7238052/
https://ncbi.nlm.nih.gov/pubmed/32295247
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/pharmaceutics12040358
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