Učitavanje...

A New Paroxetine-Based GRK2 Inhibitor Reduces Internalization of the μ-Opioid Receptor

G protein-coupled receptor (GPCR) kinases (GRKs) play a key role in terminating signals initiated by agonist-bound GPCRs. However, chronic stimulation of GPCRs, such as that which occurs during heart failure, leads to the overexpression of GRKs and maladaptive downregulation of GPCRs on the cell sur...

Cijeli opis

Spremljeno u:
Bibliografski detalji
Izdano u:Mol Pharmacol
Glavni autori: Bouley, Renee A., Weinberg, Zara Y., Waldschmidt, Helen V., Yen, Yu-Chen, Larsen, Scott D., Puthenveedu, Manojkumar A., Tesmer, John J.G.
Format: Artigo
Jezik:Inglês
Izdano: The American Society for Pharmacology and Experimental Therapeutics 2020
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC7237867/
https://ncbi.nlm.nih.gov/pubmed/32234810
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.119.118661
Oznake: Dodaj oznaku
Bez oznaka, Budi prvi tko označuje ovaj zapis!