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Validation of the Slow Off‐Kinetics of Sirtuin‐Rearranging Ligands (SirReals) by Means of Label‐Free Electrically Switchable Nanolever Technology

We have discovered the sirtuin‐rearranging ligands (SirReals) to be highly potent and selective inhibitors of the NAD(+)‐dependent lysine deacetylase Sirt2. Using a biotinylated SirReal in combination with biolayer interferometry, we previously observed a slow dissociation rate of the inhibitor–enzy...

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Detalhes bibliográficos
Publicado no:Chembiochem
Main Authors: Schiedel, Matthias, Daub, Herwin, Itzen, Aymelt, Jung, Manfred
Formato: Artigo
Idioma:Inglês
Publicado em: John Wiley and Sons Inc. 2020
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7217041/
https://ncbi.nlm.nih.gov/pubmed/31692222
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/cbic.201900527
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