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Prediction of Metabolite‐to‐Parent Drug Exposure: Derivation and Application of a Mechanistic Static Model

In the development of new drugs, the prediction of metabolite‐to‐parent plasma exposure ratio in humans prior to administration in a clinical study has emerged as an important need. In this work, we derived a mechanistic static model based on first principles to estimate metabolite‐to‐parent plasma...

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Veröffentlicht in:Clin Transl Sci
Hauptverfasser: Callegari, Ernesto, Varma, Manthena V.S., Obach, R. Scott
Format: Artigo
Sprache:Inglês
Veröffentlicht: John Wiley and Sons Inc. 2020
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC7214656/
https://ncbi.nlm.nih.gov/pubmed/31880865
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/cts.12734
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