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Design, Synthesis, and Biological Evaluation of Aromatic Amide-Substituted Benzimidazole-Derived Chalcones. The Effect of Upregulating TP53 Protein Expression

A series of benzimidazole-derived chalcones containing aromatic amide substituent were designed and synthesized. All of the chalcone compounds were tested for their in vitro antitumor activity against human cancer cell lines (HCT116, HepG2, A549, and CRL-5908). The antiproliferative activity of comp...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Argitaratua izan da:Molecules
Egile Nagusiak: Wu, Lintao, Yang, Yuting, Wang, Zhijun, Wu, Xi, Su, Feng, Li, Mengyao, Jing, Xiaobi, Han, Chun
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: MDPI 2020
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC7179225/
https://ncbi.nlm.nih.gov/pubmed/32150865
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules25051162
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