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Lasmiditan inhibits calcitonin gene-related peptide release in the rodent trigeminovascular system
Migraine headache pathophysiology involves trigeminovascular system activation, calcitonin gene-related peptide (CGRP) release, and dysfunctional nociceptive transmission. Triptans are 5-HT(1B/1D/(1F)) receptor agonists that prejunctionally inhibit trigeminal CGRP release, but their vasoconstrictor...
Tallennettuna:
| Julkaisussa: | Pain |
|---|---|
| Päätekijät: | , , , , , , , , |
| Aineistotyyppi: | Artigo |
| Kieli: | Inglês |
| Julkaistu: |
Wolters Kluwer
2020
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| Aiheet: | |
| Linkit: | https://ncbi.nlm.nih.gov/pmc/articles/PMC7170441/ https://ncbi.nlm.nih.gov/pubmed/31977930 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1097/j.pain.0000000000001801 |
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