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The radiosensitizer Onalespib increases complete remission in (177)Lu-DOTATATE-treated mice bearing neuroendocrine tumor xenografts

PURPOSE: (177)Lu-DOTATATE targeting the somatostatin receptor (SSTR) is utilized for treatment of neuroendocrine tumors (NETs). Onalespib, a heat shock protein 90 (HSP90) inhibitor, has demonstrated radiosensitizing properties and may thus enhance the effect of (177)Lu-DOTATATE. Consequently, the ai...

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Publicat a:Eur J Nucl Med Mol Imaging
Autors principals: Lundsten, Sara, Spiegelberg, Diana, Raval, Nakul R., Nestor, Marika
Format: Artigo
Idioma:Inglês
Publicat: Springer Berlin Heidelberg 2020
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7075859/
https://ncbi.nlm.nih.gov/pubmed/31912256
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s00259-019-04673-1
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