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Solid-Phase Synthesis of β-Amino Ketones Via DNA-Compatible Organocatalytic Mannich Reactions

One-bead-one-compound (OBOC) libraries constructed by solid-phase split-and-pool synthesis are a valuable source of protein ligands. Most OBOC libraries are comprised of oligoamides, particularly peptides, peptoids, and peptoid-inspired molecules. Further diversification of the chemical space covere...

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Detalhes bibliográficos
Publicado no:ACS Comb Sci
Main Authors: Tran-Hoang, Nam, Kodadek, Thomas
Formato: Artigo
Idioma:Inglês
Publicado em: 2018
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7074847/
https://ncbi.nlm.nih.gov/pubmed/29316387
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acscombsci.7b00151
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